{"product_id":"metoprolol-tartrate-for-injection-5-ml-single-dose-vials-10-box","title":"Metoprolol Tartrate Injection 5 mg\/ml Vials 10\/Box Pfizer Hospira (RX)","description":"\u003cp\u003eMetoprolol Tartrate for Injection is used primarily to manage acute episodes of hypertension and to control heart rate in patients experiencing tachycardia or other arrhythmias. It is a beta-blocker that works by blocking beta-adrenergic receptors, reducing heart rate, cardiac output, and blood pressure. This formulation is particularly useful in emergency settings, such as after a heart attack, to reduce the heart's workload and oxygen demand. Administered intravenously, it offers rapid action in stabilizing cardiac conditions.\u003c\/p\u003e\n\u003cp\u003eMetoprolol Tartrate Injection is a beta-blocker medication provided by Pfizer Injectables, intended for intravenous use. It is primarily used for the rapid control of heart rate and blood pressure in acute settings, such as during a myocardial infarction (heart attack) or to manage arrhythmias and severe hypertension. The formulation is available in single-dose vials of 5 mL, and each box contains 10 vials. \u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eDetails and Features\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eActive Ingredient:\u003c\/strong\u003e Metoprolol Tartrate\u003cbr\u003e\u003cstrong\u003eConcentration:\u003c\/strong\u003e Usually formulated to provide a specified amount of metoprolol tartrate per mL (check specific packaging for precise details).\u003cbr\u003e\u003cstrong\u003eVolume: \u003c\/strong\u003e5 mL per vial\u003cbr\u003e\u003cstrong\u003ePackaging:\u003c\/strong\u003e 10 single-dose vials per box\u003cbr\u003e\u003cstrong\u003eAdministration Route:\u003c\/strong\u003e Intravenous (IV) injection\u003cbr\u003e\u003cstrong\u003eIndications:\u003c\/strong\u003e Rapid treatment of acute myocardial infarction, control of heart rate in tachyarrhythmias (like atrial fibrillation or flutter), acute hypertension, and in certain cases, stable heart failure as adjunct therapy.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eMechanism of Action\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp\u003eMetoprolol Tartrate is a selective beta-1 adrenergic receptor blocker, primarily affecting cardiac tissues. By inhibiting the action of catecholamines (such as adrenaline) on beta-1 receptors, metoprolol reduces heart rate, cardiac output, and blood pressure. It decreases myocardial oxygen demand by lowering heart rate and contractility, which is particularly beneficial during heart attacks as it helps minimize heart muscle damage. Additionally, it can decrease electrical activity in the heart, helping to manage arrhythmias.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eWarnings\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eHeart Block and Bradycardia:\u003c\/strong\u003e Contraindicated in patients with significant bradycardia or advanced heart block unless a pacemaker is in place.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eHypotension:\u003c\/strong\u003e Use caution in patients with low blood pressure, as it can further decrease blood pressure.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eAsthma and COPD:\u003c\/strong\u003e Although selective, beta-blockers can affect beta-2 receptors at higher doses, potentially exacerbating bronchospasms in susceptible individuals.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eAcute Heart Failure:\u003c\/strong\u003e Initiation or dosage increments in acute heart failure should be done cautiously, as beta-blockers can initially cause worsening symptoms.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eAbrupt Withdrawal:\u003c\/strong\u003e Sudden discontinuation can lead to rebound tachycardia, hypertension, or even precipitate angina or myocardial infarction. Dosing should typically be tapered.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cspan style=\"text-decoration: underline;\"\u003e\u003cstrong\u003eSide Effects\u003c\/strong\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003cp\u003e\u003cem\u003eWhile metoprolol tartrate is effective, it can have side effects, especially when used acutely and intravenously:\u003c\/em\u003e\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eCommon Side Effects:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003eFatigue or lethargy\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003eDizziness or lightheadedness\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003eBradycardia (slow heart rate)\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003eHypotension\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cstrong\u003eSerious Side Effects:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003eSevere bradycardia or heart block\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003eHeart failure exacerbation\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003eBronchospasm in individuals with a history of respiratory disorders\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003eCardiogenic shock in susceptible patients\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cstrong\u003eOther Considerations:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eMonitoring: \u003c\/strong\u003eDuring administration, continuous monitoring of cardiac function (heart rate, ECG) and blood pressure is advisable. Adjustments to dose or infusion rate may be necessary based on the patient's response.\u003cbr\u003e\u003cstrong\u003eDrug Interactions:\u003c\/strong\u003e Metoprolol may interact with other medications, such as other antihypertensives, antiarrhythmics, and certain antidepressants, necessitating a comprehensive medication review.\u003c\/p\u003e\n\u003cp\u003eMetoprolol Tartrate for Injection is a potent medication used in critical care and emergency settings, offering rapid management of cardiovascular conditions when oral administration is not feasible. Its use should be overseen by healthcare professionals to ensure safe administration and effective therapeutic outcomes.\u003cbr\u003e\u003c\/p\u003e","brand":"Pfizer Injectables","offers":[{"title":"Default Title","offer_id":53337471025470,"sku":"00409-1778-05","price":2784.99,"currency_code":"INR","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0872\/3408\/5182\/files\/Metoprolol-Tartrate-Injection-5-mg-Pfizer-Hospira.jpg?v=1776771091","url":"https:\/\/himkhand.com\/products\/metoprolol-tartrate-for-injection-5-ml-single-dose-vials-10-box","provider":"Himkhand","version":"1.0","type":"link"}